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| Transmitters | |||
|---|---|---|---|
| Precursors: | None | ||
| Synthesizing enzymes: | None | ||
| Inactivation: | Reuptake Glutamate transaminase | ||
| Metabolite: | Glutamine | ||
| Receptors | |||
| Receptor types | Agonists | Antagonists | Second messenger |
| NMDA
|
NMDA, CPP, trans-2,3-PDA, (-)-cis-1-ACPD |
CGP37849 MK801: Channel blocker; PCP: Non-competitive AP5 & AP7 |
Ca++ Mg++: Voltage sensitive Glycine: Regulatory |
| AMPA:
1
2 |
AMPA, Quisqualate |
NBQX, CNQX DNQX |
Cation conductance |
| Kainate
|
Kainate, Domoate |
NBQX, CNQX DNQX |
Cation conductance |
| Metabotropic
|
1S,3R-ACPD, Ibotenate |
None | PI; G-protein |